E-Pub Full Text Articles

Benzophenone Esters and Sulfonates: Synthesis and their Potential as Antiinflammatory Agents

Author(s): Arshia, Almas Jabeen, Aisha Faheem, Khalid Mohammed Khan*, Shazia Shah and Shahnaz Perveen
Pages: 1-13 (13)
Synthesis and Evaluation of the in vitro Antimicrobial Activity of Triazoles, Morpholine and Thiosemicarbazones

Author(s): Felipe R. S. Santos, Jessica T. Andrade, Carla D. F. Sousa, Joice S. Fernandes, Lucas F. Carmo, Marcelo G. F. Araujo, Jaqueline M. S. Ferreira and Jose A. F. P. Villar*
Pages: 1-13 (13)
Synthetic Diethyl 2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylates Induce Apoptosis

Author(s): Seunghyun Ahn, Youngshim Lee, Jihyun Park, Junho Lee, Soon Young-Shin, Young Han Lee, Dongsoo Koh* and Yoongho Lim*
Pages: 1-12 (12)
4-Hydroxy-2-pyridone Derivatives and the δ-pyrone Isostere as Novel Agents Against Mycobacterium smegmatis Biofilm Inhibitors

Author(s): Maheshkumar R. Borkar, Santosh Nandan*, M N Harish Kumar , Jayashree Puttur, M Jisha , Dipankar Chatterji and Evans C. Coutinho *
Pages: 1-10 (10)
Synthesis & Anticancer Evaluation of New Substituted 2-(3,4- Dimethoxyphenyl)benzazoles

Author(s): Cigdem Karaaslan , Yalcin Duydu, Aylin Ustundag , Can Ozgur Yalcin, Banu Kaskatepe and Hakan Goker*
Pages: 1-11 (11)
Synthesis and Structural Elucidation of Novel Benzothiazole Derivatives as Anti-tubercular Agents: In-silico Screening for Possible Target Identification

Author(s): Katharigatta N. Venugopala*, Sandeep Chandrashekharappa, Melendhran Pillay, Subhrajyoti Bhandary, Mahmoud Kandeel, Fawzi M. Mahomoodally , Mohamed A. Morsy, Deepak Chopra , Bandar E. Aldhubiab, Mahesh Attimarad, Osama I. Alwassil , Sree Harsha and Koleka Mlisana
Pages: 1-16 (16)
Neuropharmacological Screening of Chiral and Non-chiral Phthalimide- Containing Compounds in Mice: in vivo and in silico Experiments

Author(s): Carolina Campos-Rodriguez, Jose G. Trujillo-Ferrara*, Ameyali Alvarez-Guerra, Iran M. Cumbres Vargas, Roberto I. Cuevas-Hernandez, Erik Andrade-Jorge, Sergio Zamudio and Eduardo Ramirez-San Juan*
Pages: 1-17 (17)
Synthesis and Biological Evaluation of Novel 2,3-disubstituted Benzofuran Analogues of GABA as Neurotropic Agents

Author(s): Arturo Coaviche-Yoval, Hector Luna, Ricardo Tovar-Miranda, Marvin Antonio Soriano-Ursua and Jose G. Trujillo-Ferrara*
Pages: 1-10 (10)
Novel Hydroxamic Acids Incorporating 1-((1H-1,2,3-Triazol-4-yl)methyl)- 3-substituted-2-oxoindolines: Synthesis, Biological Evaluation and SAR Analysis

Author(s): Do Thi Mai Dung, Nguyen Van Huan, Do Manh Cam, Dao Cam Hieu, Pham-The Hai, Le-Thi-Thu Huong, Jisung Kim, Jeong Eun Choi, Jong Soon Kang, Sang-Bae Han* and Nguyen-Hai Nam*
Pages: 1-20 (20)
The Evaluation of Metal Co-ordinating Bis-Thiosemicarbazones as Potential Anti-malarial Agents

Author(s): Fady N. Akladios, Scott D. Andrew, Samantha J. Boog, Carmen de Kock, Richard K. Haynes and Christopher J. Parkinson*
Pages: 1-8 (8)
2-Oxo-1,2,3,4-tetrahydropyrimidines as Potent β-Glucuronidase Inhibitors: One-pot Synthesis, In vitro and In silico Studies

Author(s): Sarosh Iqbal*, Nimra Naveed Shaikh, Khalid Mohammed Khan*, Sehrish Naz, Zaheer Ul-Haq Qasmi, Shahnaz Perveen and M. Iqbal Choudhary*
Pages: 1-12 (12)
Pyrano[3,2-c]quinoline Derivatives as New Class of α-glucosidase Inhibitors to Treat Type 2 Diabetes: Synthesis, in vitro Biological Evaluation and Kinetic Study

Author(s): Zahra Heydari, Maryam Mohammadi-Khanaposhtani, Somaye Imanparast, Mohammad Ali Faramarzi, Mohammad Mahdavi *, Parviz Rashidi Ranjbar* and Bagher Larijani
Pages: 1-9 (9)
Homopiperazine Derived Female Controlled Vaginal Trichomonacidal Contraceptive: An Addition to Structure-Activity Relationship

Author(s): B. S. Rahul , Bindu Saraswati, C. Shiju, Gopal Gupta and Nand Lal*
Pages: 1-11 (11)
Design, Synthesis and Biological Evaluation of 1H-1,2,3-Triazole-Linked- 1H

Author(s): Carolina S. Bortolot, Luana da S. M. Forezi, Roberta K. F. Marra, Marcelo I. P. Reis, Barbara V. F. e Sa, Ricardo Imbroisi Filho, Zeinab Ghasemishahrestani, Mauro Sola-Penna, Patricia Zancan, Vitor F. Ferreira* and Fernando de C. da Silva*
Pages: 1-11 (11)
Design, Synthesis and Investigation of New Diphenyl Substituted Pyridazinone Derivatives as Both Cholinesterase and Aβ-Aggregation Inhibitors

Author(s): Burcu Kilic, Merve Erdogan, Hayrettin O. Gulcan, Fatma Aksakal, Nihan Oruklu, E. Umit Bagriacik and Deniz S. Dogruer*
Pages: 1-18 (18)
Exploration of (hetero)aryl Derived Thienylchalcones for Antiviral and Anticancer Activities

Author(s): Vikrant Patil, Siddappa A. Patil*, Renukadevi Patil, Alejandro Bugarin, Kenneth Beaman and Shivaputra A. Patil*
Pages: 1-12 (12)
Antimicrobial Evaluation of Erythrinan Alkaloids from Erythrina cristagalli L.

Author(s): Janaina M. de Avila, Ionara I. Dalcol*, Alessandra O. Pereira, Eveline W. Santos, Adriano Ferraz, Maura Z. Santos, Marco Aurelio Mostardeiro and Ademir F. Morel
Pages: 1-7 (7)
Sorbinil, an Aldolase Reductase Inhibitor, in Fighting Against Diabetic Complications

Author(s): Qi Huang, Qiong Liu and Dongsheng Ouyang*
Pages: 1-5 (5)
Synthesis of Nucleosides and Non-nucleosides Based 4,6-disubstituted-2- oxo-dihydropyridine-3-carbonitriles as Antiviral Agents

Author(s): Tarek S. Ibrahim, Hassan A. El-Sayed, Maan T. Khayat, Amany M.M. AL-Mahmoudy, Ahmed H. Moustafa, Ayat K. Saad El-Deen, Sherif A.F. Rostom and Siva S. Panda*
Pages: 1-18 (18)
Crystal Structure of Mistletoe Lectin I (ML-I) from Viscum album in Complex with 4-N-Furfurylcytosine at 2.85 Å Resolution

Author(s): Malik Shoaib Ahmad*, Saima Rasheed, Sven Falke, Binish Khaliq, Markus Perbandt, M. Iqbal Choudhary, Wojciech T. Markiewicz, Jan Barciszewski and Christian Betzel*
Pages: 1-10 (10)
Pyrazole and imidazo[1,2-b]pyrazole Derivatives as New Potential Antituberculosis Agents

Author(s): Elda Meta, Chiara Brullo*, Michele Tonelli, Scott G. Franzblau, Yuehong Wang, Rui Ma, Wan Baojie , Beatrice Silvia Orena, Maria Rosalia Pasca and Olga Bruno
Pages: 1-11 (11)
Synthesis and Biological Evaluation of 12N-substituted Tricyclic Matrinic Derivatives as a Novel Family of Anti-Influenza Agents

Author(s): Sheng Tang, Yu-Huan Li , Xin–Yue Cheng, Jin–Qiu Yin , Ying–Hong Li , Dan–Qing Song , Yan–Xiang Wang * and Zhan–Dong Liu
Pages: 1-9 (9)
Identification of New Chromenone Derivatives as Cholinesterase Inhibitors and Molecular Docking Studies

Author(s): Jamshed Iqbal *, Muhammad Shakeel Ahmad Abbasi, Sumera Zaib , Saifullah Afridi, Norbert Furtmann, Jurgen Bajorath and Peter Langer
Pages: 1-9 (9)

E-Pub Full Text Articles

Benzophenone Esters and Sulfonates: Synthesis and their Potential as Antiinflammatory Agents

Synthesis and Evaluation of the in vitro Antimicrobial Activity of Triazoles, Morpholine and Thiosemicarbazones

Synthetic Diethyl 2,6-dimethyl-1,4-dihydropyridine-3,5-dicarboxylates Induce Apoptosis

4-Hydroxy-2-pyridone Derivatives and the δ-pyrone Isostere as Novel Agents Against Mycobacterium smegmatis Biofilm Inhibitors

Synthesis & Anticancer Evaluation of New Substituted 2-(3,4- Dimethoxyphenyl)benzazoles

Synthesis and Structural Elucidation of Novel Benzothiazole Derivatives as Anti-tubercular Agents: In-silico Screening for Possible Target Identification

Neuropharmacological Screening of Chiral and Non-chiral Phthalimide- Containing Compounds in Mice: in vivo and in silico Experiments

Synthesis and Biological Evaluation of Novel 2,3-disubstituted Benzofuran Analogues of GABA as Neurotropic Agents

Novel Hydroxamic Acids Incorporating 1-((1H-1,2,3-Triazol-4-yl)methyl)- 3-substituted-2-oxoindolines: Synthesis, Biological Evaluation and SAR Analysis

The Evaluation of Metal Co-ordinating Bis-Thiosemicarbazones as Potential Anti-malarial Agents

2-Oxo-1,2,3,4-tetrahydropyrimidines as Potent β-Glucuronidase Inhibitors: One-pot Synthesis, In vitro and In silico Studies

Pyrano[3,2-c]quinoline Derivatives as New Class of α-glucosidase Inhibitors to Treat Type 2 Diabetes: Synthesis, in vitro Biological Evaluation and Kinetic Study

Homopiperazine Derived Female Controlled Vaginal Trichomonacidal Contraceptive: An Addition to Structure-Activity Relationship

Design, Synthesis and Biological Evaluation of 1H-1,2,3-Triazole-Linked- 1H

Design, Synthesis and Investigation of New Diphenyl Substituted Pyridazinone Derivatives as Both Cholinesterase and Aβ-Aggregation Inhibitors

Exploration of (hetero)aryl Derived Thienylchalcones for Antiviral and Anticancer Activities

Antimicrobial Evaluation of Erythrinan Alkaloids from Erythrina cristagalli L.

Sorbinil, an Aldolase Reductase Inhibitor, in Fighting Against Diabetic Complications

Synthesis of Nucleosides and Non-nucleosides Based 4,6-disubstituted-2- oxo-dihydropyridine-3-carbonitriles as Antiviral Agents

Crystal Structure of Mistletoe Lectin I (ML-I) from Viscum album in Complex with 4-N-Furfurylcytosine at 2.85 Å Resolution

Pyrazole and imidazo[1,2-b]pyrazole Derivatives as New Potential Antituberculosis Agents

Synthesis and Biological Evaluation of 12N-substituted Tricyclic Matrinic Derivatives as a Novel Family of Anti-Influenza Agents

Identification of New Chromenone Derivatives as Cholinesterase Inhibitors and Molecular Docking Studies